Compound index
Filter by tier, goal, or class — or search by name. Each profile carries regulatory status, mechanism, and every human study we could verify.
74 compounds
Afamelanotide (MT-I) / Melanotan II
MC1R (pigment), MC3/4R.
Bremelanotide (PT-141)
MC4R agonist.
Collagen peptides
Hydrolysate di/tripeptides.
Elamipretide (SS-31)
Binds inner mitochondrial membrane cardiolipin.
Estradiol / Progesterone (menopause HRT)
ER/PR agonists.
Gonadorelin & GnRH analogs
GnRH agonists (leuprolide, triptorelin, goserelin) cause downregulation; antagonists (degarelix, relugolix, elagolix) block directly.
hCG
LH-receptor agonist.
Insulin (incl. bodybuilding misuse)
Insulin receptor agonist.
Liraglutide
Daily GLP-1RA; t½ ~13 h.
Octreotide / Lanreotide
SSTR2/5 agonists.
Orforglipron
Small-molecule GLP-1R agonist, once-daily oral without food restriction.
Oxytocin
OXTR agonist.
Pramlintide
Amylin agonist.
Semaglutide
GLP-1R agonist; t½ ~7 d (SC weekly); oral formulation with SNAC.
Setmelanotide
MC4R agonist.
Somatropin (recombinant HGH)
GH receptor agonist.
Teriparatide / Abaloparatide
PTH1R anabolic.
Tesamorelin
Stabilized GHRH(1-44).
Testosterone (all esters, TRT)
AR agonist; esters (cypionate, enanthate, undecanoate), gels, pellets, oral TU.
Thyroid hormone (T4/T3)
TR agonists.
Tirzepatide
Dual GIP/GLP-1R agonist; t½ ~5 d.
Vosoritide
NPR-B agonist.
Anastrozole & other AIs
Block aromatase.
BPC-157
Proposed NO/VEGF/growth-factor effects; rodent data.
Clomiphene / Enclomiphene
Hypothalamic ER antagonism ↑LH/FSH.
DHEA / Pregnenolone
Precursors to androgens/estrogens/neurosteroids.
Nandrolone & other AAS
AR agonist (19-nortestosterone).
Sermorelin
GHRH-R agonist, t½ minutes.
Actovegin (deproteinized calf-blood hemodialysate)
Origin: Austria/Russia (Takeda, later others); widely used in Russia/E.
Amycretin
Unimolecular GLP-1/amylin agonist.
AOD-9604
Claimed lipolytic fragment.
Bromantane (Ladasten) [NEW, sport]
Origin: Russia.
Cagrilintide / CagriSema
Amylin/calcitonin receptor agonist, weekly.
Cerebrolysin
Neurotrophic mixture.
Chinese GLP-1 agonists: beinaglutide, PEG-loxenatide [NEW split]
Origin: China.
CJC-1295
Albumin-binding GHRH; t½ ~6-8 d.
Cortexin (Кортексин)
Polypeptide fraction from cerebral cortex of livestock; claimed neuroprotective.
Cycloferon (meglumine acridonacetate)
Low-molecular-weight interferon inducer (non-peptide).
Dalargin (Даларгин)
Synthetic Leu-enkephalin analog Tyr-D-Ala-Gly-Phe-Leu-Arg.
Dihexa
HGF/c-Met potentiator.
Ecdysterone (20-hydroxyecdysone) [NEW, sport]
Origin: USSR-origin research (Leuzea/Rhaponticum); global supplement.
Efpeglenatide (Korea, Hanmi) [NEW, replaces Korea placeholder]
Origin: South Korea.
Epitalon
Claimed telomerase activation.
GHK-Cu
Copper-binding tripeptide; collagen synthesis in vitro.
GHRP-2 / GHRP-6 / Hexarelin
GHS-R1a agonists.
Heberprot-P (recombinant human EGF) — Cuba
Origin: Cuba (CIGB).
Humanin
Cytoprotective mitokine.
IGF-1 LR3 / Mecasermin
IGF-1R agonist.
Imunofan (Arg-α-Asp-Lys-Val-Tyr-Arg) [NEW]
Synthetic hexapeptide (thymopoietin fragment-derived) immunomodulator 1.
Ipamorelin
Selective GHS-R1a agonist.
Khavinson short peptides (Cytogens/'peptide bioregulators': Pinealon EDR, Vilon KE, Livagen, etc.)
Hypothesis that di-/tripeptides enter cells and bind histones/DNA to alter gene expression.
Kisspeptin
KISS1R → GnRH.
KPV
NF-κB anti-inflammatory.
LL-37
Antimicrobial/immunomodulatory.
Mazdutide
Glucagon/GLP-1 dual agonist.
Meldonium (Mildronate) [NEW, sport]
Inhibits carnitine biosynthesis → reduced β-oxidation, shift to glycolysis; anti-ischemic 2.
Mexidol (emoxypine succinate)
3-hydroxypyridine antioxidant (non-peptide).
MK-677 (ibutamoren) — non-peptide
Oral ghrelin mimetic; t½ ~24 h.
MOTS-c
AMPK activation.
Noopept (omberacetam, GVS-111)
N-phenylacetyl-L-prolylglycine ethyl ester (dipeptide-derived).
Oral-Turinabol (4-chlorodehydromethyltestosterone) — GDR history [NEW, sport]
Origin: East Germany (VEB Jenapharm).
Oxandrolone
Oral AAS.
Phenibut (β-phenyl-GABA)
GABA-B (some GABA-A) agonist, baclofen analog 1.
Phenylpiracetam (fonturacetam, Phenotropil, carphedon)
Origin: Russia.
Retatrutide
Triple agonist; t½ ~6 d.
SARMs (ostarine, LGD-4033, RAD-140)
Tissue-selective AR agonists.
Selank (Селанк, Thr-Lys-Pro-Arg-Pro-Gly-Pro)
Tuftsin analog / ACTH(4-10) analog.
Semax (Семакс, Met-Glu-His-Phe-Pro-Gly-Pro)
Tuftsin analog / ACTH(4-10) analog.
Survodutide
Glucagon/GLP-1 dual agonist.
TB-500 / Thymosin β4
Tβ4 sequesters G-actin; TB-500 = LKKTETQ fragment.
Thymalin (Тималин)
Polypeptide complex extracted from bovine thymus; immunomodulator (T-cell function).
Thymogen (Тимоген, α-Glu-Trp)
Synthetic dipeptide alpha-glutamyl-tryptophan (immunomodulator derived from thymalin research).
Thymosin α1
T-cell maturation, TLR signaling.
Trimetazidine [NEW, sport]
Origin: France origin; heavy use in Russia/E.